Found 421 recordings
DICL IDIon ChannelCompound FunctionSpeciesValueReferences
DICL_CP_0307708Glutamate receptor ionotropic subunit kainate 1AntagonistHomo sapiens (Human)Ki: 118 nM10.1124/mol.53.2.195, 9463476
DICL_CP_0307823Glutamate receptor ionotropic subunit kainate 1ModulatorHomo sapiens (Human)Ki: 701 nM10.1016/s0028-3908(98)00122-1, 9849663
DICL_CP_0307837Glutamate receptor ionotropic subunit kainate 1InhibitorHomo sapiens (Human)Ki: 140 nM10.1021/jm800092x, 18578478
DICL_CP_0307844Glutamate receptor ionotropic subunit kainate 1AgonistHomo sapiens (Human)EC50: 130000 nM10.1021/jm701394a, 18338843
DICL_CP_0307846Ionotropic glutamate receptor (Glutamate receptor 5)AgonistHomo sapiens (Human)EC50: 130000 nM10.1021/jm701394a, 18338843
DICL_CP_0307858Glutamate receptor ionotropic subunit kainate 1AntagonistHomo sapiens (Human)Ki: 140 nM10.1021/jm301433m, 23414088
DICL_CP_0307865Glutamate receptor ionotropic subunit kainate 1AgonistHomo sapiens (Human)EC50: 83500 nM10.1021/jm2004078, 21619066
DICL_CP_0307866Glutamate receptor ionotropic subunit kainate 1AgonistHomo sapiens (Human)EC50: 35200 nM10.1016/s0960-894x(00)00346-2, 10969973
DICL_CP_0307867Glutamate receptor 5AgonistHomo sapiens (Human)EC50: 75000 nM10.1016/s0960-894x(00)00346-2, 10969973
DICL_CP_0307874Glutamate receptor ionotropic subunit kainate 1AgonistHomo sapiens (Human)EC50: 140000 nM10.1021/jm900565c, 19588945
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